SCHEMBL1383207

SCHEMBL1383207

[NH]C(=O)C(c1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
HDAC3 O15379 1/20 0.54
HDAC4 P56524 1/20 0.54
HDAC1 Q13547 1/20 0.54
HDAC7 Q8WUI4 1/20 0.54
HDAC2 Q92769 1/20 0.54
HDAC10 Q969S8 1/20 0.54
HDAC11 Q96DB2 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
HDAC6 Q9UBN7 1/20 0.54
HDAC9 Q9UKV0 1/20 0.54
HDAC5 Q9UQL6 1/20 0.54
CTSD P07339 1/20 0.52
CYP2D6 P10635 1/20 0.50
POLB P06746 1/20 0.50
SRC P12931 1/20 0.50
LMNA P02545 3/20 0.48
MAPK1 P28482 1/20 0.48
CES2 O00748 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylacetic Acid SCHEMBL8513250 0.78 SRC (0.62) TDP1L3MBTL1HDAC3HDAC4HDAC1
Diphenylacetic Acid SCHEMBL38022 0.78 SRC (0.62) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL465969 0.78 TDP1 (0.61) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL3728852 0.77 LMNA (0.65) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL11223553 0.77 SRC (0.48) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL4849143 0.77 LMNA (0.65) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL4850637 0.77 LMNA (0.65) TDP1L3MBTL1HDAC3HDAC4HDAC1
SCHEMBL7450800 0.77 TDP1 (0.43) TDP1L3MBTL1HDAC3HDAC4HDAC1
Diphenylacetic Acid SCHEMBL6852183 0.76 SRC (0.59) TDP1L3MBTL1HDAC3HDAC4HDAC1
Diphenylacetic Acid SCHEMBL8411440 0.76 SRC (0.59) TDP1L3MBTL1HDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 94 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337536-B1 CATIONIC GROUP-3 CATALYST SYSTEM EXXONMOBIL CHEM PATENTS INC (US) 2012-09-12 EP claimed
JP-4838934-B2 2011-12-14 JP claimed
US-7390861-B2 Cationic group-3 catalyst system EXXONMOBIL CHEMICAL PATENTS INC. (US) 2008-06-24 US claimed
EP-1044197-B1 PIPERIDINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKYNE CARBOXAMIDES AS CYTOSTATIC AGENTS AND IMMUNOSUPPRESSANTS ASTELLAS PHARMA GMBH (DE) 2006-04-19 EP claimed
EP-1042291-B1 ARYL-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS KLINGE CO CHEM PHARM FAB (DE) 2005-07-13 EP claimed
EP-1515997-A1 YTTRIUM-BASED ETHYLENE POLYMERIZATION CATALYSTS WITH BULKY AMIDINATE ANCILLARY LIGANDS ExxonMobil Chemical Patents Inc. (US) 2005-03-23 EP claimed
US-20040033889-A1 Yttrium-based ethylene polymerization catalysts with bulky amidinate ancillary ligands EXXONMOBIL CHEMICAL PATENTS INC. 2004-02-19 US claimed
US-20040033891-A1 Cationic group-3 catalyst system EXXONMOBIL CHEMICAL PATENTS INC. 2004-02-19 US claimed
WO-2004000894-A1 YTTRIUM-BASED ETHYLENE POLYMERIZATION CATALYSTS WITH BULKY AMIDINATE ANCILLARY LIGANDS EXXONMOBIL CHEMICAL PATENTS INC. (US) 2003-12-31 WO claimed
EP-1337536-A1 CATIONIC GROUP-3 CATALYST SYSTEM ExxonMobil Chemical Patents Inc. (US) 2003-08-27 EP claimed
US-6593344-B1 These substances have especially high cytostatic activities and pronounced immunosuppressive properties which make them suitable for therapeutic treatment in broad tumor spectrum and autoimmune diseases KLINGE PHARMA GMBH (DE) 2003-07-15 US claimed
WO-2002032909-A1 CATIONIC GROUP-3 CATALYST SYSTEM EXXONMOBIL CHEMICAL PATENTS INC. (US) 2002-04-25 WO claimed
EP-1044197-A2 NEW PIPERIDINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES Klinge Pharma GmbH (DE) 2000-10-18 EP claimed
EP-1042291-A1 ARYL-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS Klinge Pharma GmbH (DE) 2000-10-11 EP claimed
WO-1999031060-A2 PIPERIDINYL-SUBSTITUTED PYRIDYLALKANE, ALKENE AND ALKINE CARBOXAMIDES AS CYTOSTATICS AND IMMUNESUPPRESSANTS KLINGE PHARMA GMBH (DE) 1999-06-24 WO claimed
WO-1999031064-A1 ARYL-SUBSTITUTED PYRIDYLALKANE, ALKENE, AND ALKINE CARBOXAMIDES USEFUL AS CYTOSTATIC AND IMMUNOSUPPRESSIVE AGENTS KLINGE PHARMA GMBH (DE) 1999-06-24 WO claimed
EP-0552489-B1 Peptide, production and use thereof TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1998-03-04 EP claimed
US-10077288-B2 Hydroxystatin derivatives for the treatment of arthrosis MERCK PATENT GMBH (DE) 2018-09-18 US disclosed
US-4151300-A CENTRAL NERVOUS SYSTEM, PSYCHOTROPIC LABORATOIRE L. LAFON (FR) 1979-04-24 US disclosed
US-4122186-A PSYCHOTROPIC AGENTS LABORATOIRE L. LAFON (FR) 1978-10-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10077288-B2 Hydroxystatin derivatives for the treatment of arthrosis CTSD, CTSB, CTSZ TDP1 1632/4885L3MBTL1 2640/4885HDAC3 766/4885
US-20040033891-A1 Cationic group-3 catalyst system COG3, ORC3, LIG3 TDP1 4378/4885L3MBTL1 489/4885HDAC3 816/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.