SCHEMBL7450860

SCHEMBL7450860

Brc1cncc(OCc2ccccc2)c1.Oc1cncc(Br)c1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 5/20 0.54
LMNA P02545 1/20 0.47
CYP1A2 P05177 1/20 0.47
PTGS1 P23219 1/20 0.47
SLC6A2 P23975 1/20 0.47
CYP2C19 P33261 1/20 0.47
PTGS2 P35354 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HIF1A Q16665 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
PTGES O14684 1/20 0.43
P4HTM Q9NXG6 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX5 P09917 1/20 0.41
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL188660 0.92 MAOB (0.62) MAOBLMNACYP1A2PTGS1SLC6A2
SCHEMBL6582384 0.88 CYP1A2 (0.56) MAOBLMNACYP1A2PTGS1SLC6A2
SCHEMBL6933324 0.85 MAOB (0.47) MAOBSMN1; SMN2
SCHEMBL24619909 0.81 LTA4H (0.51) MAOB
SCHEMBL8512404 0.81 MAOB (0.56) MAOBLMNACYP1A2PTGS1SLC6A2
SCHEMBL31418062 0.78 MAOB (0.64) MAOBLMNACYP1A2PTGS1SLC6A2
SCHEMBL9369289 0.78 RAB9A (0.49) MAOBALOX5
SCHEMBL21675841 0.77 MAOB (0.62) MAOB
SCHEMBL6119008 0.77 MAOB (0.68) MAOB
SCHEMBL189829 0.76 MAOB (0.53) MAOBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147112-A1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2001-10-24 EP disclosed
WO-2000044755-A1 DIAZABICYCLIC DERIVATIVES AS NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS ABBOTT LABORATORIES (US) 2000-08-03 WO disclosed