SCHEMBL7452863

SCHEMBL7452863

Nc1ccc(NCC(O)CO)c(-c2cc[nH]c2)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
CHEK1 O14757 1/20 0.31
CDK1 P06493 1/20 0.31
AR P10275 1/20 0.30
VDR P11473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7461982 0.88
SCHEMBL6574847 0.85 PDE3B (0.37) PDE3BPDE3ACHEK1CDK1AR
SCHEMBL6572042 0.84 PDE3B (0.34) PDE3BPDE3ACHEK1CDK1AR
SCHEMBL6571461 0.82 CHEK1 (0.41) CHEK1CDK1
SCHEMBL6573407 0.81 USP7 (0.36) PDE3BPDE3AARVDR
Hydrochloric Acid SCHEMBL6572537 0.81 CHEK1 (0.40) CHEK1CDK1
SCHEMBL7462106 0.81 PRSS1 (0.32)
SCHEMBL6571859 0.81 KDM4E (0.37) CHEK1CDK1
SCHEMBL6571878 0.80 CYP1A2 (0.38) PDE3BPDE3A
SCHEMBL6571824 0.80 CYP1A2 (0.34) PDE3BPDE3AARVDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0963982-B1 New diaminobenzene derivatives and these componends containing colouring agents WELLA AG (DE) 2002-03-13 EP disclosed
US-6132475-A FOR OXIDATION DYEING OF KERATIN FIBERS; INCLUDES COUPLER AND DEVELOPER, IN WHICH THE DEVELOPER IS A SUBSTITUTED 2-(FURYL, THIENYL, PYRROLYL, OR SELENOPHENE) P-DIAMINOBENZENE DERIVATIVE OF GIVEN FORMULA; COLORFASTNESS, WASHFASTNESS WELLA AKTIENGESELLSCHAFT (DE) 2000-10-17 US disclosed
EP-0963982-A2 New diaminobenzene derivatives and these componends containing colouring agents Wella Aktiengesellschaft (DE) 1999-12-15 EP disclosed