SCHEMBL7454479

SCHEMBL7454479

N#CCCCCCCl.N#CCCCCCl

nearest known ligand 0.56

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.56
CYP3A4 P08684 1/20 0.56
ALDH1A1 P00352 3/20 0.41
TDP1 Q9NUW8 2/20 0.41
MAPT P10636 1/20 0.37
LOX P28300 1/20 0.33
LOXL3 P58215 1/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
HIF1A Q16665 2/20 0.31
EPAS1 Q99814 2/20 0.31
GBA1 P04062 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11225741 1.00
SCHEMBL14351852 1.00 TSHR (0.56) TSHRCYP3A4ALDH1A1TDP1MAPT
SCHEMBL850797 1.00
SCHEMBL851045 0.97
SCHEMBL435492 0.87
SCHEMBL25030516 0.85 TSHR (0.42) TSHRCYP3A4ALDH1A1TDP1MAPT
SCHEMBL10532870 0.85 TSHR (0.42) TSHRCYP3A4ALDH1A1TDP1MAPT
Bicarbonate SCHEMBL11778367 0.84 TSHR (0.46) TSHRCYP3A4ALDH1A1TDP1MAPT
SCHEMBL1003333 0.83 ALDH1A1 (0.58) TSHRCYP3A4ALDH1A1TDP1MAPT
SCHEMBL818520 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1030665-A4 THERAPEUTIC USES OF QUINOLINE DERIVATIVES AVENTIS PHARM PROD INC (US) 2002-11-27 EP disclosed
EP-1030665-A1 THERAPEUTIC USES OF QUINOLINE DERIVATIVES Aventis Pharmaceuticals Products Inc. (US) 2000-08-30 EP disclosed
WO-1999020275-A1 THERAPEUTIC USES OF QUINOLINE DERIVATIVES AVENTIS PHARMACEUTICALS PRODUCTS INC. (US) 1999-04-29 WO disclosed
EP-0397697-A4 QUINOLINE DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4? 1991-07-03 EP disclosed
EP-0397697-A1 QUINOLINE DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D 4?. RORER INT OVERSEAS (US) 1990-11-22 EP disclosed
WO-1989004304-A1 QUINOLINE DERIVATIVES AS ANTAGONISTS OF LEUKOTRIENE D4 RORER INTERNATIONAL (OVERSEAS) INC. (US) 1989-05-18 WO disclosed