SCHEMBL7455141

SCHEMBL7455141

O[C@H](CBr)c1ccc(Cl)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 1/20 0.50
TP53 P04637 2/20 0.47
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
KCNH2 Q12809 2/20 0.43
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GRIN2B Q13224 2/20 0.39
NPSR1 Q6W5P4 2/20 0.38
IDO1 P14902 2/20 0.38
TDO2 P48775 1/20 0.38
TOP2A P11388 1/20 0.37
TOP2B Q02880 1/20 0.37
MITF O75030 1/20 0.36
MAPT P10636 1/20 0.36
XBP1 P17861 1/20 0.36
MAPK1 P28482 1/20 0.36
NTSR1 P30989 1/20 0.36
KMT2A Q03164 1/20 0.36
PAX8 Q06710 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7786053 1.00 ADRA2C (0.50) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL30514270 1.00 ADRA2C (0.50) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL7783863 0.82 TSHR (0.36) ADRA2CLMNAHTTTSHRMAPT
SCHEMBL11452909 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL7460986 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL3124491 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL7453698 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL6212874 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL10396657 0.82 LMNA (0.53) ADRA2CTP53LMNAHTTKCNH2
SCHEMBL29845931 0.82 ADRA2C (0.51) ADRA2CTP53LMNAHTTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017108972-A1 COMPOUNDS OF R-(-)-(E)-[4-(2,4-DICHLOROPHENYL)-1,3-DITHIOLAN-2-YLIDENE]-1 -IMIDAZOLYLACETONITRILE-HA (LULICONAZOLE-HA) AS ANTIFUNGALS LABORATORIOS LESVI, S.L. (ES) 2017-06-29 WO disclosed
WO-2017108972-A1 COMPOUNDS OF R-(-)-(E)-[4-(2,4-DICHLOROPHENYL)-1,3-DITHIOLAN-2-YLIDENE]-1 -IMIDAZOLYLACETONITRILE-HA (LULICONAZOLE-HA) AS ANTIFUNGALS LABORATORIOS LESVI, S.L. (ES) 2017-06-29 WO disclosed
CN-106008166-A Industrialized production method of chiral 2- chloro-1-(2,4-dichlorophenyl) ethanol 上海福乐医药科技有限公司 2016-10-12 CN disclosed
EP-0839035-B1 ANTIFUNGAL AGENT, COMPOUND THEREFOR, PROCESS FOR PRODUCING THE SAME NIHON NOHYAKU CO LTD (JP) 2002-10-02 EP disclosed
US-5900488-A Method for treating mycosis using imidazolylacetonitrile derivatives NIHON NOHYAKU CO., LTD. (JP) 1999-05-04 US disclosed
EP-0839035-A2 ANTIFUNGAL AGENT, COMPOUND THEREFOR, PROCESS FOR PRODUCING THE SAME Nihon Nohyaku Co., Ltd. (JP) 1998-05-06 EP disclosed
WO-1997002821-A2 ANTIFUNGAL AGENT, COMPOUND THEREFOR, PROCESS FOR PRODUCING THE SAME NIHON NOHYAKU CO., LTD. (JP) 1997-01-30 WO disclosed