SCHEMBL745516

SCHEMBL745516

CC(C)(C)c1ccc(CN(CCCc2ccc(Cl)c(Cl)c2)C(=O)c2cc(Cl)cc3c2NCCC3)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
LMNA P02545 2/20 0.35
HSP90AA1 P07900 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
NR1H4 Q96RI1 1/20 0.32
ESRRB O95718 1/20 0.32
ESRRG P62508 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
TACR2 P21452 1/20 0.32
TACR1 P25103 1/20 0.32
MAPT P10636 1/20 0.32
SIGMAR1 Q99720 5/20 0.32
LPAR1 Q92633 3/20 0.32
LPAR2 Q9HBW0 1/20 0.32
TRPV1 Q8NER1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL746670 0.99 PARP1 (0.35) PARP1LMNAHSP90AA1PSEN1PSEN2
SCHEMBL745512 0.96 OPRM1 (0.34) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL747110 0.95 OPRM1 (0.34) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL751012 0.89 PARP1 (0.36) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL747122 0.88 TP53 (0.33) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL747648 0.88 PARP1 (0.36) PARP1PSEN1PSEN2APH1BNCSTN
SCHEMBL746654 0.88 OPRM1 (0.34) PARP1HSP90AA1NR1H4ESRRBESRRG
Hydrochloric Acid SCHEMBL748492 0.88 TP53 (0.33) PARP1PSEN1PSEN2APH1BNCSTN
Hydrochloric Acid SCHEMBL751441 0.87 OPRM1 (0.33) PARP1HSP90AA1NR1H4ESRRBESRRG
SCHEMBL746554 0.87 TP53 (0.34) NR1H4ESRRBESRRGTACR2TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed