SCHEMBL746654

SCHEMBL746654

Cc1cc2c(c(C(=O)N(CCc3ccc(Cl)c(Cl)c3)Cc3ccc(C(C)(C)C)cc3)c1)NCCC2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
TRPV1 Q8NER1 1/20 0.33
HSP90AA1 P07900 1/20 0.33
SIGMAR1 Q99720 8/20 0.32
TP53 P04637 3/20 0.32
CYP1A2 P05177 3/20 0.32
ESRRG P62508 2/20 0.32
CYP2D6 P10635 2/20 0.32
TSHR P16473 2/20 0.32
NR1H4 Q96RI1 1/20 0.32
ESRRB O95718 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
CYP3A4 P08684 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL751441 0.99 OPRM1 (0.33) OPRM1OPRD1CRHBPCRHR2TRPV1
SCHEMBL745512 0.92 OPRM1 (0.34) OPRM1OPRD1CRHBPCRHR2SIGMAR1
Hydrochloric Acid SCHEMBL747110 0.92 OPRM1 (0.34) OPRM1OPRD1CRHBPCRHR2SIGMAR1
SCHEMBL746554 0.91 TP53 (0.34) OPRM1OPRD1SIGMAR1TP53CYP1A2
Hydrochloric Acid SCHEMBL748806 0.90 TP53 (0.33) OPRM1OPRD1SIGMAR1TP53CYP1A2
SCHEMBL745501 0.89 TMEM97 (0.39) OPRM1OPRD1CRHBPCRHR2SIGMAR1
SCHEMBL745516 0.88 PARP1 (0.35) OPRM1OPRD1TRPV1HSP90AA1SIGMAR1
Hydrochloric Acid SCHEMBL752637 0.88 TMEM97 (0.38) OPRM1OPRD1CRHBPCRHR2SIGMAR1
SCHEMBL748282 0.88 TP53 (0.39) CRHBPCRHR2TRPV1TP53ESRRG
Hydrochloric Acid SCHEMBL746670 0.87 PARP1 (0.35) OPRM1OPRD1TRPV1HSP90AA1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US claimed
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed