SCHEMBL7455503

SCHEMBL7455503

O=C1NC(=O)C(S(=O)(=O)c2ccccc2F)S1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.40
AKR1B1 P15121 1/20 0.37
HSD11B1 P28845 4/20 0.36
MAPT P10636 2/20 0.36
GBA1 P04062 1/20 0.35
KMT2A Q03164 2/20 0.35
PPARG P37231 1/20 0.35
KAT6A Q92794 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
PTGER3 P43115 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303679 0.77 CA2 (0.49) CA2MAPTPPARGL3MBTL1NPSR1
SCHEMBL8651760 0.74 CDK2 (0.37) CA2MAPTKMT2ANPSR1KDM4E
SCHEMBL8302470 0.71 CA2 (0.39) CA2MAPTKMT2APPARGKAT6A
SCHEMBL144642 0.70 LMNA (0.47) CA2AKR1B1L3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL8647686 0.69 AKR1B1 (0.37) AKR1B1KMT2AKAT6AL3MBTL1NPSR1
SCHEMBL6784875 0.68 F2 (0.39) CA2MAPT
SCHEMBL6754040 0.68 ALDH1A1 (0.43) CA2MAPTKMT2ASMN1; SMN2ALDH1A1
SCHEMBL8303252 0.68 MAPT (0.41) CA2MAPTKMT2APPARGNPSR1
SCHEMBL8647785 0.66 MAPT (0.42) CA2MAPTKMT2ANPSR1KDM4E
SCHEMBL8304958 0.66 GAA (0.36) CA2MAPTKMT2AL3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804193-A4 THIAZOLIDINE DERIVATIVES FOR THE TREATMENT OF PSORIASIS KURTZ THEODORE W (US) 2002-03-27 EP disclosed
US-5824694-A Thiazolidine derivatives for the treatment of psoriasis BETHESDA PHARMACEUTICALS, INC. (US) 1998-10-20 US disclosed
EP-0804193-A1 THIAZOLIDINE DERIVATIVES FOR THE TREATMENT OF PSORIASIS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-11-05 EP disclosed
US-5594015-A Thiazolidine derivatives for the treatment of psoriasis REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-01-14 US disclosed
WO-1995035108-A1 THIAZOLIDINE DERIVATIVES FOR THE TREATMENT OF PSORIASIS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-28 WO disclosed