SCHEMBL7457052

SCHEMBL7457052

COC(=O)C(C)Oc1ccc(C)c(-c2nsc3ccc(-n4c(=O)cc(C)n(C)c4=O)cc23)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
ALDH2 P05091 1/20 0.36
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
MAPT P10636 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KLK7 P49862 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7457042 0.86 PABPC1 (0.33) POLBSMN1; SMN2L3MBTL1
SCHEMBL7463638 0.84 POLB (0.35) POLBSMN1; SMN2ALDH2
SCHEMBL7461699 0.84 POLB (0.36) POLBSMN1; SMN2ALDH2MEN1KMT2A
SCHEMBL7456892 0.83
SCHEMBL7468039 0.83 KDM4E (0.39) MEN1KMT2AKDM4EALDH1A1HPGD
SCHEMBL7463298 0.83
SCHEMBL7452381 0.82 PPARD (0.36) KDM4EALDH1A1HPGD
SCHEMBL7460387 0.81 LMNA (0.30) LMNATP53
SCHEMBL7462525 0.81 TAS1R3 (0.32)
SCHEMBL7464741 0.80

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed