SCHEMBL7459184

SCHEMBL7459184

Cc1ccc(OCC(=O)N(C(C)C)C(C)C)c(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)c1

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.31
ACHE P22303 1/20 0.31
MEN1 O00255 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31
SRD5A2 P31213 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453077 0.91 TRPM8 (0.33) BCHEACHE
SCHEMBL7461736 0.91 PTGDR2 (0.31)
SCHEMBL7459566 0.90 PTGDR2 (0.38) MEN1KMT2A
SCHEMBL7051566 0.89 KDM4E (0.35) MEN1KMT2A
SCHEMBL7455498 0.88 ALPL (0.33)
SCHEMBL7459199 0.88 PPARD (0.33) BCHEACHEMEN1TSHRKMT2A
SCHEMBL7460136 0.87 MEN1 (0.33) MEN1KMT2A
SCHEMBL7462824 0.87 TP53 (0.33)
SCHEMBL7467239 0.87 PTGDR2 (0.34)
SCHEMBL8339743 0.85 ESR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed