SCHEMBL7459199

SCHEMBL7459199

Cc1cc(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)ccc1OCC(=O)N(C(C)C)C(C)C

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 16/20 0.33
PPARA Q07869 6/20 0.33
BCHE P06276 1/20 0.33
ACHE P22303 1/20 0.33
SRD5A2 P31213 2/20 0.32
PPARG P37231 2/20 0.32
MEN1 O00255 1/20 0.31
TSHR P16473 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7453085 0.91 PPARD (0.33) PPARDPPARABCHEACHEPPARG
SCHEMBL7455505 0.88 OXTR (0.36) PPARDPPARAMEN1KMT2A
SCHEMBL7459184 0.88 BCHE (0.31) BCHEACHESRD5A2MEN1TSHR
SCHEMBL7453732 0.85 ALDH1A1 (0.33)
SCHEMBL7458904 0.84 PTGS2 (0.36)
SCHEMBL7463328 0.84 KDM4E (0.31)
SCHEMBL7461757 0.84
SCHEMBL7457864 0.84
SCHEMBL7457226 0.82 HPGD (0.43) MEN1KMT2A
SCHEMBL7456944 0.82

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed