SCHEMBL7459476

SCHEMBL7459476

Fc1c[c]ccc1Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.43
HTR2A P28223 1/20 0.41
CALM1 P0DP23 1/20 0.41
BCL2 P10415 1/20 0.39
BCL2L1 Q07817 1/20 0.39
LTA4H P09960 1/20 0.38
CTRC Q99895 3/20 0.36
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
PTPN1 P18031 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9561120 0.85 HTR2A (0.41) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL2094181 0.82 CALM1 (0.46) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL8210180 0.77 BCL2 (0.53) ALOX5CALM1BCL2BCL2L1HPGD
SCHEMBL7453249 0.77 CALM1 (0.41) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL7465412 0.77 CALM1 (0.41) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL27920117 0.77 HTR2A (0.41) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL8939761 0.77 KDM4E (0.37) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL28651733 0.76 TAAR1 (0.43) HTR2AKMT2APTPN1
SCHEMBL29130603 0.76 CALM1 (0.39) ALOX5HTR2ACALM1BCL2BCL2L1
SCHEMBL1584544 0.76 LMNA (0.40) HTR2AKMT2APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209453-A Methylene linked quinolinyl modulators of ROR-gamma-T JANSSEN PHARMACEUTICA NV 2015-12-30 CN disclosed
EP-1140900-A4 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY INC (US) 2002-04-10 EP disclosed
EP-1140900-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2001-10-10 EP disclosed
WO-2000039083-A2 PYRAZOLE COMPOUNDS AND USES THEREOF PPD DISCOVERY, INC. (US) 2000-07-06 WO disclosed