SCHEMBL7459587

SCHEMBL7459587

Clc1cccc(-c2[c]ccc(-c3ccccc3)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.44
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
TSHR P16473 1/20 0.42
NFKB1 P19838 1/20 0.42
RAB9A P51151 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX5 P09917 1/20 0.42
MAOB P27338 2/20 0.41
PGR P06401 4/20 0.40
CYP1A2 P05177 1/20 0.39
ESR2 Q92731 1/20 0.39
SCN2A Q99250 1/20 0.38
IDO1 P14902 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GABRP O00591 1/20 0.36
GABRD O14764 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3022644 0.85 ALOX5 (0.42) TAAR1NPC1TP53TSHRNFKB1
SCHEMBL7222040 0.83 TAAR1 (0.44) TAAR1ALOX5MAOBPGRESR2
SCHEMBL1451004 0.82 ALDH1A1 (0.43) TAAR1ALOX5CYP1A2ESR2
SCHEMBL8938017 0.81 ALOX5 (0.41) TAAR1NPC1RAB9ASMN1; SMN2ALOX5
SCHEMBL15067523 0.80 ALDH1A1 (0.45) TAAR1ALOX5CYP1A2ESR2
SCHEMBL1535844 0.80 ALDH1A1 (0.38) NPC1RAB9AALOX5ESR2
SCHEMBL7470031 0.80 ADORA2A (0.43) PGRCYP1A2ESR2ADORA2AADORA1
SCHEMBL29788033 0.80 TAAR1 (0.61) TAAR1NPC1TP53TSHRNFKB1
SCHEMBL170231 0.80 TAAR1 (0.61) TAAR1NPC1TP53TSHRNFKB1
SCHEMBL27998968 0.80 ALOX5 (0.43) TAAR1NPC1TP53TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed