SCHEMBL7459606

SCHEMBL7459606

COC(=O)c1c(C(F)(F)F)[nH]c2c(O)cc3c(c12)C(CCl)CN3C(=O)c1cc2cc(NC(=O)c3cc4ccccc4cn3)ccc2[nH]1

nearest known ligand 0.32

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.32
SRC P12931 1/20 0.32
SYK P43405 4/20 0.32
ABCB1 P08183 3/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 3/20 0.31
RAB9A P51151 3/20 0.31
ALDH1A1 P00352 1/20 0.31
PRNP P04156 1/20 0.31
GAA P10253 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PYGL P06737 1/20 0.31
BRD4 O60885 1/20 0.31
ADH1A P07327 1/20 0.30
KIT P10721 1/20 0.30
FLT1 P17948 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30
ABL2 P42684 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463782 0.95 ABL1 (0.32) ABL1SRCSYKABCB1ABCG2
SCHEMBL7469597 0.93 PYGL (0.32) SYKNPC1RAB9APYGLADH1A
SCHEMBL7468222 0.91 NPC1 (0.37) ABCB1KDM4ENPC1RAB9AALDH1A1
SCHEMBL7460674 0.91 GABRA1 (0.37) KDM4ENPC1RAB9AALDH1A1GABRA1
SCHEMBL7460322 0.91 BRAF (0.36) ABL1SRCSYKABCB1ABCG2
SCHEMBL7473460 0.90 ABCB1 (0.35) ABCB1KDM4ENPC1RAB9APYGL
SCHEMBL7463553 0.89 KDM4E (0.36) SYKKDM4ENPC1RAB9AALDH1A1
SCHEMBL7458517 0.89 P4HB (0.34) ABCB1KDM4ENPC1RAB9AALDH1A1
SCHEMBL8831163 0.89 P4HB (0.34) ABCB1KDM4ENPC1RAB9AALDH1A1
SCHEMBL7460763 0.89 KDM4E (0.37) SYKKDM4ENPC1RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0656360-B1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2002-11-20 EP disclosed
US-5629430-A ANTICARCINOGENIC AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-05-13 US disclosed
EP-0656360-A1 TRIFLUOROMETHYLPYRROLOINDOLE CARBOXYLIC ESTER DERIVATIVE AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1995-06-07 EP disclosed