SCHEMBL7459783

SCHEMBL7459783

COC(=O)c1c(Cl)cc(Cl)cc1NC(=O)CSc1ccc(O)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
CYP1A2 P05177 4/20 0.53
CYP2C9 P11712 4/20 0.53
CYP2C19 P33261 4/20 0.53
CYP2D6 P10635 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 4/20 0.50
KDM4E B2RXH2 3/20 0.50
HTT P42858 2/20 0.50
GAA P10253 2/20 0.50
KMT2A Q03164 2/20 0.50
MAPT P10636 2/20 0.49
CYP3A4 P08684 3/20 0.47
HPGD P15428 1/20 0.47
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
TP53 P04637 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462894 0.90 KDM4E (0.64) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7461619 0.90 ALDH1A1 (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7461299 0.85 KMT2A (0.53) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7459046 0.83 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7467908 0.82 RAB9A (0.53) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7463414 0.82 L3MBTL1 (0.60) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7467237 0.82 KDM4E (0.52) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7462314 0.82 MAPT (0.59) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7456883 0.81 ALDH1A1 (0.53) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6
SCHEMBL7456897 0.81 KMT2A (0.48) ALDH1A1CYP1A2CYP2C9CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0869122-B1 Quinolinic sulfide derivatives acting as NMDA receptor antagonists and process for preparation thereof KOREA RES INST CHEM TECH (KR) 2002-12-04 EP disclosed
US-5990126-A 4-HYDROXY-QUINOLIN-2-ONE DERIVATIVES SUBSTITUTED AT POSITION 3 WITH A SUBSTITUTED AROMATIC- OR HETEROAROMATIC-SULFIDE GROUP; ANTAGONIST OF EXCITATORY AMINO ACID FOR NMDA RECEPTORS; TREATING EPILEPSY, STROKE, PARKINSON'S DISEASE KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1999-11-23 US disclosed
EP-0869122-A1 Quinolinic sulfide derivatives acting as NMDA receptor antagonists and process for preparation thereof KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1998-10-07 EP disclosed