SCHEMBL7460629

SCHEMBL7460629

O=C=Nc1ccc2c(c1)OC(CC(F)(F)F)(C(F)(F)F)O2

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CYP3A4 P08684 2/20 0.34
TSHR P16473 1/20 0.34
TRPA1 O75762 1/20 0.34
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11003249 0.77 MAPK1 (0.43) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL10451237 0.77 MAPK1 (0.43) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL10645022 0.73 MAPK1 (0.47) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL7470763 0.72 AHR (0.39) TSHR
SCHEMBL7462347 0.72 PDK2 (0.36) CYP3A4CYP1A2
SCHEMBL11002226 0.67 MAPK1 (0.37) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL592019 0.63 ADRA2A (0.53) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL29648863 0.63 HTR3E (0.53) MAPK1TDP1CYP3A4TRPA1
SCHEMBL29540837 0.63 ADRA2A (0.53) MAPK1TDP1CYP3A4TSHRTRPA1
SCHEMBL140824 0.63 HTR3E (0.53) MAPK1TDP1CYP3A4TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0596359-B1 Fluorinated 1,3-benzo- and 1,3-pyrido-dioxoles, process for their preparation and their use for the preparation of plant-protective agents BAYER AG (DE) 2002-07-03 EP disclosed
US-5482956-A ANTIPROTOZOA AGENTS FOR ANIMALS OR INSECTS BAYER AKTIENGESELLSCHAFT (DE) 1996-01-09 US disclosed
US-5420309-A Plant saftening agents, insecticides or nematocides BAYER AKTIENGESELLSCHAFT (DE) 1995-05-30 US disclosed
EP-0597304-A1 Use of substituted benzimidazoles BAYER AG (DE) 1994-05-18 EP disclosed
EP-0596359-A2 Fluorinated 1,3-benzo- and 1,3-pyrido-dioxoles, process for their preparation and their use for the preparation of plant-protective agents BAYER AG (DE) 1994-05-11 EP disclosed