SCHEMBL7461682

SCHEMBL7461682

CC(C)N(CCCCCN1C(=O)COc2ccccc21)C(C)C

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMPD1 P17405 1/20 0.53
CHRM1 P11229 5/20 0.51
POLB P06746 1/20 0.51
HSD17B10 Q99714 1/20 0.51
DRD2 P14416 3/20 0.50
HTR2A P28223 3/20 0.50
MCHR1 Q99705 2/20 0.50
F2 P00734 1/20 0.49
F10 P00742 1/20 0.49
PRSS1 P07477 1/20 0.49
ALOX12 P18054 1/20 0.47
ALDH1A1 P00352 1/20 0.47
HTR1A P08908 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
TSHR P16473 1/20 0.46
DRD4 P21917 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15423257 0.82 POLB (0.55) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL15423258 0.82 DRD2 (0.56) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL10248078 0.81 POLB (0.56) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL764345 0.80 POLB (0.55) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL16264966 0.79 DRD2 (0.58) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL1764705 0.79 ALDH1A1 (0.55) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL13618147 0.78 DRD2 (0.61) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL1763884 0.78 DRD2 (0.57) SMPD1CHRM1DRD2HTR2AMCHR1
SCHEMBL4058329 0.77 ALDH1A1 (0.56) SMPD1CHRM1POLBHSD17B10DRD2
SCHEMBL318658 0.76 TSHR (0.58) SMPD1CHRM1POLBHSD17B10DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1068191-A1 BENZOXAZINONES/BENZOTHIAZINONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2001-01-17 EP disclosed
WO-1999050257-A1 BENZOXAZINONES/BENZOTHIAZINONES AS SERINE PROTEASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1999-10-07 WO disclosed