SCHEMBL7463111

SCHEMBL7463111

Cc1nccn1-c1nc(-c2ccc(Cl)cc2)c(CCC=O)o1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
RXRA P19793 3/20 0.33
RXRB P28702 3/20 0.33
RXRG P48443 3/20 0.33
MAPKAPK2 P49137 3/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
BRD4 O60885 1/20 0.32
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
KCNH2 Q12809 2/20 0.31
GPR142 Q7Z601 2/20 0.31
CACNA1C Q13936 1/20 0.31
SCN5A Q14524 1/20 0.31
SMN1; SMN2 Q16637 3/20 0.30
KDM4E B2RXH2 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460783 0.85 MAPKAPK2 (0.35) ALDH1A1RXRARXRBRXRGMAPKAPK2
SCHEMBL6606347 0.84 RXRA (0.47) ALDH1A1RXRARXRBRXRGSMN1; SMN2
SCHEMBL963990 0.83 SIRT2 (0.40) ALDH1A1RXRARXRBRXRGMAPKAPK2
SCHEMBL7463531 0.83 MAPKAPK2 (0.34) ALDH1A1MAPKAPK2PSEN1PSEN2APH1B
SCHEMBL7462674 0.83 NR4A2 (0.37) RXRARXRBRXRGMAPKAPK2CYP3A4
SCHEMBL965656 0.83 SIRT2 (0.37) ALDH1A1RXRARXRBRXRGMAPKAPK2
SCHEMBL7456651 0.83 ALDH1A1 (0.34) ALDH1A1MAPKAPK2CYP3A4CYP2D6KCNH2
SCHEMBL7461461 0.82 RXRA (0.43) RXRARXRBRXRG
SCHEMBL1360344 0.82 SIRT2 (0.36) RXRARXRBRXRGMAPKAPK2CYP3A4
SCHEMBL964061 0.82 SIRT2 (0.36) RXRARXRBRXRGMAPKAPK2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891340-B1 OXAZOLE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-11-13 EP disclosed