SCHEMBL7464371

SCHEMBL7464371

O=C(O)c1ccc(Cl)cc1NCc1ccncc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
GRIK1 P39086 2/20 0.59
L3MBTL1 Q9Y468 1/20 0.59
KDM4C Q9H3R0 7/20 0.56
KDM4E B2RXH2 3/20 0.56
KDM6B O15054 1/20 0.56
KDM4A O75164 1/20 0.56
KDM4D Q6B0I6 1/20 0.56
ACLY P53396 1/20 0.53
CDC7 O00311 1/20 0.52
ROCK2 O75116 1/20 0.52
MAP4K4 O95819 1/20 0.52
GSK3B P49841 1/20 0.52
CLK4 Q9HAZ1 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
HTT P42858 1/20 0.51
KDM5B Q9UGL1 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
ALDH1A1 P00352 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688887 0.87 ACLY (0.64) MEN1KMT2AGRIK1L3MBTL1KDM4C
SCHEMBL7467939 0.84 GRIK1 (0.59) GRIK1KDM4CKDM4EKDM6BKDM4A
SCHEMBL1714812 0.83 KDM4C (0.56) MEN1KMT2AL3MBTL1KDM4CKDM4E
SCHEMBL4980301 0.83 KDR (0.64) HDAC1KDRMAPK1
SCHEMBL15817727 0.80 KDM4C (0.76) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL1715089 0.79 KDM4C (0.70) MEN1KMT2AL3MBTL1KDM4CKDM4E
SCHEMBL1714819 0.79 KDM4C (0.85) KDM4CKDM4EKDM6BKDM4AKDM4D
SCHEMBL14389304 0.78 ACLY (0.51) MEN1KMT2AGRIK1KDM4EACLY
SCHEMBL29855520 0.78 ACLY (0.51) MEN1KMT2AGRIK1KDM4EACLY
SCHEMBL7461503 0.77 HPGD (0.60) MEN1KMT2AGRIK1KDM4EACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed