SCHEMBL7464402

SCHEMBL7464402

N[C@@H](CNC(=O)c1cccc(N2CCC(Nc3ncccn3)CC2)c1)C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.44
CNR2 P34972 3/20 0.44
DRD2 P14416 5/20 0.42
DRD3 P35462 5/20 0.42
ITGB3 P05106 2/20 0.41
ITGA2B P08514 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2C Q14957 2/20 0.41
TLR2 O60603 2/20 0.41
HDAC1 Q13547 1/20 0.40
ITGAV P06756 1/20 0.40
PDGFRB P09619 1/20 0.40
KDR P35968 1/20 0.40
EPHX2 P34913 1/20 0.39
PRMT5 O14744 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28747046 0.89 ITGB3 (0.49) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL382962 0.89 ITGB3 (0.49) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL6499974 0.85 ITGB3 (0.43) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL6496378 0.84 ITGB3 (0.42) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL382676 0.84 ITGB3 (0.52) ITGB3ITGA2BGRIN3BGRIN1GRIN2C
SCHEMBL6500046 0.83 PRMT5 (0.44) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL7464438 0.83 DRD2 (0.42) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL6499934 0.82 ITGB3 (0.61) ITGB3ITGA2BITGAV
SCHEMBL6503934 0.82 ITGB3 (0.42) CNR1CNR2DRD2DRD3ITGB3
SCHEMBL382099 0.82 ITGB3 (0.54) DRD2DRD3ITGB3ITGA2BGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP claimed
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP disclosed