SCHEMBL7464438

SCHEMBL7464438

NC(CC(=O)O)NC(=O)c1cccc(N2CCC(Nc3ncccn3)CC2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 6/20 0.42
DRD3 P35462 6/20 0.42
CNR1 P21554 4/20 0.41
CNR2 P34972 3/20 0.41
HDAC1 Q13547 1/20 0.40
P2RY12 Q9H244 1/20 0.38
KDR P35968 1/20 0.38
SCN9A Q15858 1/20 0.38
VCP P55072 1/20 0.38
PLOD2 O00469 2/20 0.38
PLOD3 O60568 2/20 0.38
PLOD1 Q02809 2/20 0.38
CASR P41180 1/20 0.38
EPHX2 P34913 1/20 0.38
ITGB3 P05106 1/20 0.37
ITGB1 P05556 1/20 0.37
ITGAV P06756 1/20 0.37
ITGA2B P08514 1/20 0.37
ITGA5 P08648 1/20 0.37
ITGB5 P18084 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL382964 0.89 CASR (0.45) DRD2DRD3HDAC1CASREPHX2
SCHEMBL6500015 0.86 DRD2 (0.40) DRD2DRD3CNR1CNR2HDAC1
SCHEMBL382678 0.84 ITGB3 (0.44) EPHX2ITGB3ITGAVITGA2B
SCHEMBL7464402 0.83 CNR1 (0.44) DRD2DRD3CNR1CNR2HDAC1
SCHEMBL6499964 0.82 KAT6A (0.43) DRD2DRD3CNR1CNR2HDAC1
SCHEMBL382101 0.82 ITGB3 (0.46) DRD2DRD3CASRITGB3ITGAV
SCHEMBL6501602 0.81 KDM4E (0.56) DRD2DRD3CNR1CNR2PLOD2
SCHEMBL7467089 0.81 ITGB3 (0.43) DRD2DRD3VCPITGB3ITGAV
SCHEMBL6507021 0.80 ITGB3 (0.41) DRD2DRD3CNR1CNR2ITGB3
SCHEMBL6496356 0.80 HDAC1 (0.41) DRD2DRD3CNR1CNR2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP claimed
EP-1229024-A1 m-SUBSTITUTED BENZOIC ACID DERIVATIVES EXHIBITING INTEGRIN ALPHA-V BETA-3 ANTAGONISM MEIJI SEIKA KAISHA LTD. (JP) 2002-08-07 EP disclosed