SCHEMBL7464574

SCHEMBL7464574

Cc1cccc(C=C2NC(=O)SC2=O)c1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 8/20 0.68
PIM2 Q9P1W9 8/20 0.68
CSNK2A2 P19784 1/20 0.55
CLK1 P49759 1/20 0.55
CSNK2B P67870 1/20 0.55
CSNK2A1 P68400 1/20 0.55
DYRK1A Q13627 1/20 0.55
DYRK2 Q92630 1/20 0.55
DYRK1B Q9Y463 1/20 0.55
NAT1 P18440 1/20 0.54
AKR1B1 P15121 4/20 0.46
GSK3B P49841 1/20 0.46
CISD1 Q9NZ45 3/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
HPGD P15428 1/20 0.45
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
TTR P02766 1/20 0.43
PIM3 Q86V86 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463867 0.83 PIM1 (0.68) PIM1PIM2CSNK2A2CLK1CSNK2B
SCHEMBL2539680 0.81 PIM1 (1.00) PIM1PIM2NAT1AKR1B1GSK3B
SCHEMBL2539679 0.81 PIM1 (1.00) PIM1PIM2NAT1AKR1B1GSK3B
SCHEMBL2539676 0.81 PIM1 (1.00) PIM1PIM2NAT1AKR1B1GSK3B
SCHEMBL7465312 0.81 CSNK2A2 (0.51) PIM1PIM2CSNK2A2CLK1CSNK2B
SCHEMBL7459912 0.81 GSK3B (0.71) PIM1PIM2CSNK2A2CLK1CSNK2B
SCHEMBL7466029 0.81 CSNK2A1 (0.71) PIM1PIM2CSNK2A2CLK1CSNK2B
SCHEMBL4156417 0.80 CSNK2A2 (0.65) PIM1PIM2CSNK2A2CLK1CSNK2B
SCHEMBL3787295 0.77 IGF1R (0.71) CSNK2A2CLK1CSNK2BCSNK2A1DYRK1A
SCHEMBL7466320 0.75 PIM1 (0.73) PIM1PIM2CSNK2A2CLK1CSNK2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214305-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION Maxia Pharmaceuticals, Inc. (US) 2002-06-19 EP claimed
WO-2001016123-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION MAXIA PHARMACEUTICALS, INC. (US) 2001-03-08 WO claimed