SCHEMBL7464635

SCHEMBL7464635

Nc1nccc(NC(=O)Cn2c(=O)n(S(=O)(=O)c3ccc(Cl)cc3)c(=O)c3ccc(Cl)cc32)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.37
MAPT P10636 3/20 0.36
TP53 P04637 2/20 0.36
HRH4 Q9H3N8 2/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
S1PR2 O95136 1/20 0.35
POLB P06746 1/20 0.35
PDE5A O76074 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
RXFP1 Q9HBX9 1/20 0.34
NOD1 Q9Y239 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465244 0.87 F10 (0.43) CMA1MAPTTP53MEN1KMT2A
SCHEMBL7463810 0.86 SMN1; SMN2 (0.45) TP53MEN1KMT2AS1PR2PSEN1
SCHEMBL7472833 0.82 MAPT (0.48) CMA1MAPTTP53MEN1KMT2A
SCHEMBL7468103 0.82 GAA (0.44) CMA1MAPTTP53MEN1KMT2A
SCHEMBL7563746 0.80 MAPT (0.49) MAPTTP53MEN1KMT2AS1PR2
SCHEMBL7468006 0.79 MAPT (0.46) CMA1MAPTTP53MEN1KMT2A
SCHEMBL7468043 0.79 MAPT (0.48) MAPTTP53MEN1KMT2APOLB
SCHEMBL7463225 0.79 CMA1 (0.42) CMA1MAPTTP53S1PR2PSEN1
SCHEMBL7461911 0.79 MAPT (0.44) CMA1MAPTTP53MEN1KMT2A
SCHEMBL7466453 0.78 CMA1 (0.37) CMA1MAPTTP53S1PR2PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed