SCHEMBL7464656

SCHEMBL7464656

FC(F)(F)c1ccc(Br)c2occc12.Oc1cc(C(F)(F)F)ccc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.36
HTR2C P28335 1/20 0.34
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
XBP1 P17861 1/20 0.34
XDH P47989 1/20 0.33
SLC22A12 Q96S37 1/20 0.33
CASP3 P42574 2/20 0.33
CSNK2A2 P19784 1/20 0.32
CSNK2B P67870 1/20 0.32
CSNK2A1 P68400 1/20 0.32
AKR1C3 P42330 1/20 0.31
TMPRSS4 Q9NRS4 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
TAS2R14 Q9NYV8 1/20 0.30
CYP1A2 P05177 1/20 0.30
HSP90AA1 P07900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5987754 0.84 HTR2C (0.43) HTR2CMAPTCASP3NOTUM
SCHEMBL1928764 0.77 MEN1 (0.44) CES2MAPTNPSR1XBP1MEN1
SCHEMBL4995601 0.69 IDO1 (0.33) HTR2CCSNK2A1ALOX15
SCHEMBL6167848 0.68 HTR2C (0.31) HTR2C
SCHEMBL2001354 0.68 CES2 (0.55) CES2MAPTNPSR1TMPRSS4MEN1
SCHEMBL25193520 0.66 NLRP3 (0.38) XDHSLC22A12CASP3TSHR
SCHEMBL28171587 0.66 HTR2C (0.43) HTR2CMAPT
SCHEMBL29632676 0.65 MAPT (0.53) CES2MAPTNPSR1XBP1MEN1
SCHEMBL496276 0.65 MAPT (0.53) CES2MAPTNPSR1XBP1MEN1
SCHEMBL290533 0.65 CES2 (0.50) CES2MAPTNPSR1XBP1TAS2R14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204658-A1 BENZOFURYLPIPERAZINE SEROTONIN AGONISTS ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2001009123-A1 BENZOFURYLPIPERAZINE SEROTONIN AGONISTS ELI LILLY AND COMPANY (US) 2001-02-08 WO disclosed