SCHEMBL7465003

SCHEMBL7465003

CN1CCN(c2nccnc2OCCOc2cccnc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 2/20 0.54
CHRNB2 P17787 6/20 0.51
CHRNA4 P43681 6/20 0.51
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
CHRNA1 P02708 1/20 0.44
CHRNB1 P11230 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNB3 Q05901 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473337 0.87 HRH4 (0.50) HRH4TSHRHSD17B10
SCHEMBL4320113 0.85 CHRNB2 (0.48) CHRNB2CHRNA4CHRNA1CHRNB1CHRNB4
SCHEMBL4320526 0.76 CHRNB2 (0.44) CHRNB2CHRNA4CYP3A4CHRNA1CHRNB1
SCHEMBL4320521 0.76 CHRNB2 (0.44) CHRNB2CHRNA4CYP3A4CHRNA1CHRNB1
SCHEMBL7474070 0.76 CHRNB2 (0.44) CHRNB2CHRNA4CYP3A4CHRNA1CHRNB1
SCHEMBL15307685 0.75 CHRNB2 (0.49) CHRNB2CHRNA4ALDH1A1CYP1A2CYP3A4
SCHEMBL4310871 0.74 MAPK1 (0.48) HRH4ALDH1A1CYP1A2TSHRHSD17B10
SCHEMBL4315272 0.74 CHRNB2 (0.44) HRH4CHRNB2CHRNA4CYP1A2CYP3A4
SCHEMBL2641453 0.74 CHRNA7 (0.44) CHRNB2CHRNA4CHRNA7
SCHEMBL235730 0.74 CHRNA7 (0.44) CHRNB2CHRNA4CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1178973-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION Pharmacia AB (SE) 2002-02-13 EP disclosed
WO-2000076984-A2 NOVEL COMPOUNDS, THEIR USE AND PREPARATION BIOVITRUM AB (SE) 2000-12-21 WO disclosed