SCHEMBL7465137

SCHEMBL7465137

CC(C)(C)OC(=O)C(O)Cc1cccc(N)c1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 1/20 0.47
ADRB2 P07550 6/20 0.41
ADRB1 P08588 2/20 0.41
ADRB3 P13945 2/20 0.41
KLK5 Q9Y337 2/20 0.40
ITGA4 P13612 1/20 0.38
ITGB7 P26010 1/20 0.38
CTSS P25774 3/20 0.37
CTSK P43235 3/20 0.37
CTSB P07858 2/20 0.37
CTSL P07711 1/20 0.37
MAOA P21397 2/20 0.37
MAOB P27338 2/20 0.37
CPN1 P15169 1/20 0.36
CPB2 Q96IY4 1/20 0.36
CYP19A1 P11511 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27525604 0.86 SLC7A5 (0.56) SLC7A5ADRB2ADRB1ADRB3KLK5
SCHEMBL22442929 0.82 ADRB2 (0.40) SLC7A5ADRB2ADRB1ADRB3KLK5
SCHEMBL30759366 0.82 ITGA4 (0.51) SLC7A5KLK5ITGA4ITGB7CTSS
SCHEMBL487422 0.82 ITGA4 (0.51) SLC7A5KLK5ITGA4ITGB7CTSS
SCHEMBL487423 0.82 ITGA4 (0.51) SLC7A5KLK5ITGA4ITGB7CTSS
SCHEMBL7470063 0.81 SLC7A5 (0.46) SLC7A5ADRB2ADRB1ADRB3KLK5
SCHEMBL31689508 0.80 CTSS (0.54) KLK5CTSSCTSKCTSBCTSL
SCHEMBL3073448 0.77 CTSS (0.47) SLC7A5ADRB2KLK5CTSSCTSK
SCHEMBL755879 0.77 KDM6B (0.54) SLC7A5ADRB2MAOAMAOBCPN1
SCHEMBL6680700 0.77 KLK5 (0.61) KLK5CTSSCTSKCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6479531-B1 Gastrin and cholecystokinin receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 2002-11-12 US disclosed
EP-1178969-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2002-02-13 EP disclosed
WO-2000027823-A1 GASTRIN AND CHOLECYSTOKININ RECEPTOR LIGANDS JAMES BLACK FOUNDATION LIMITED (GB) 2000-05-18 WO disclosed