SCHEMBL7465175

SCHEMBL7465175

O=CNCC(CCCN1CCN(C(c2ccccc2)c2ccccc2)CC1)(c1ccccc1)c1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 8/20 0.51
DRD2 P14416 7/20 0.51
HRH1 P35367 5/20 0.48
KCNH2 Q12809 3/20 0.48
HRH2 P25021 2/20 0.48
HTR2A P28223 2/20 0.48
HTR2B P41595 2/20 0.48
USP2 O75604 2/20 0.48
SLC6A2 P23975 1/20 0.48
SLC6A4 P31645 1/20 0.48
SLC6A3 Q01959 1/20 0.48
TEK Q02763 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
OPRK1 P41145 2/20 0.47
ABCB11 O95342 1/20 0.47
CHRM2 P08172 1/20 0.47
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
DRD4 P21917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459803 0.85 CHRM4 (0.50) DRD3DRD2KCNH2HTR2ADRD4
Hydrochloric Acid SCHEMBL8869803 0.84 CHRM4 (0.52) DRD3DRD2KCNH2HTR2ADRD4
Hydrochloric Acid SCHEMBL7467316 0.84 CHRM4 (0.52) DRD3DRD2KCNH2HTR2ADRD4
SCHEMBL7462064 0.81 MCHR1 (0.54) CCR3
SCHEMBL7462282 0.80 DRD2 (0.49) DRD3DRD2HRH1HTR2AHTR2B
Hydrochloric Acid SCHEMBL7458878 0.80 MCHR1 (0.54) CCR3
Hydrochloric Acid SCHEMBL7459710 0.80 DRD2 (0.49) DRD3DRD2HRH1HTR2AHTR2B
SCHEMBL7464640 0.80 MCHR1 (0.53) DRD2ADRA2ACCR3
Hydrochloric Acid SCHEMBL7465064 0.79 MCHR1 (0.52) DRD2ADRA2ACCR3
SCHEMBL7464621 0.78 CCR3 (0.72) CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1219294-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP claimed
EP-1219294-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP disclosed
EP-0712845-B1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2001-10-17 EP disclosed
US-5633248-A GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS, DIARYLALKYLIDENEDIAMINES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-05-27 US disclosed
EP-0712845-A1 Amine compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-05-22 EP disclosed