SCHEMBL746527

SCHEMBL746527

O=S(=O)(CC1CCC1)N1CCC2(CCN(c3ccc(OC(F)(F)F)cc3)C2)CC1

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 4/20 0.43
FFAR4 Q5NUL3 9/20 0.41
EPHX2 P34913 3/20 0.41
DRD3 P35462 1/20 0.41
CHRM4 P08173 2/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
MMP12 P39900 1/20 0.38
MMP13 P45452 1/20 0.38
MMP14 P50281 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3737858 0.80 LIPE (0.60) LIPE
SCHEMBL745454 0.80 CYP1A2 (0.54) LIPEEPHX2
SCHEMBL743295 0.78 LIPE (0.43) LIPEFFAR4EPHX2CHRM4
SCHEMBL5888 0.75 EPHX2 (0.49) LIPEFFAR4EPHX2DRD3
SCHEMBL745746 0.74 CYP3A4 (0.58)
SCHEMBL744430 0.74 LIPE (0.68) LIPEEPHX2
SCHEMBL746672 0.74 CYP3A4 (0.73)
SCHEMBL26552871 0.73 ALDH1A1 (0.47) EPHX2MMP13MMP14
SCHEMBL764042 0.71 CYP3A4 (0.52) LIPE
SCHEMBL747836 0.71 EPHX2 (0.49) EPHX2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2430023-A1 AZACYCLIC SPIRODERIVATIVES AS HSL INHIBITORS F. Hoffmann-La Roche AG (CH) 2012-03-21 EP disclosed