SCHEMBL7465357

SCHEMBL7465357

BrCc1ccc2ccsc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.46
MRGPRX4 Q96LA9 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRK1 P41145 1/20 0.36
SIGMAR1 Q99720 1/20 0.32
TRPA1 O75762 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
PTPRC P08575 1/20 0.31
PTPN6 P29350 1/20 0.31
PTPN11 Q06124 1/20 0.31
PTPN22 Q9Y2R2 1/20 0.31
DYRK1A Q13627 1/20 0.31
PTGER4 P35408 1/20 0.31
PTGER3 P43115 1/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
CTNNB1 P35222 1/20 0.30
WNT3A P56704 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6734063 0.93 CYP2A6 (0.41) CYP2A6MRGPRX4OPRM1OPRK1PTGER4
SCHEMBL1863293 0.83 CYP2A6 (0.66) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1
SCHEMBL29469368 0.83 CYP2A6 (0.66) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1
SCHEMBL10230281 0.79 CYP2A6 (0.46) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1
SCHEMBL3150204 0.79 CYP2A6 (0.46) CYP2A6MRGPRX4OPRM1OPRK1PTPRC
SCHEMBL8058490 0.79 CYP2A6 (0.46) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1
SCHEMBL507426 0.79 CYP2A6 (0.71) CYP2A6MRGPRX4OPRM1OPRK1DYRK1A
SCHEMBL154793 0.79 CYP2A6 (0.47) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1
SCHEMBL6399446 0.78 CYP2A6 (0.54) CYP2A6OPRM1OPRK1SIGMAR1PTPRC
SCHEMBL3799097 0.76 CYP2A6 (0.43) CYP2A6MRGPRX4OPRM1OPRK1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244616-A1 (HETERO)BICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES SmithKline Beecham plc (GB) 2002-10-02 EP disclosed
WO-2001047874-A1 (HETERO)BICYCLYMETHANESULFONYLAMINO-SUBSTITUTED HYDROXAMIC ACID DERIVATIVES SMITHKLINE BEECHAM P.L.C. (GB) 2001-07-05 WO disclosed