SCHEMBL7465742

SCHEMBL7465742

CNc1cccc(OCc2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)c1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.33
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
MCHR1 Q99705 6/20 0.32
MAPT P10636 1/20 0.32
HTR2C P28335 1/20 0.31
BLK P51451 1/20 0.30
BMX P51813 1/20 0.30
JAK3 P52333 1/20 0.30
BTK Q06187 1/20 0.30
F10 P00742 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7454228 0.89 MAOB (0.43) MAOAMAOBMCHR1MAPTHTR2C
SCHEMBL7459577 0.89 MAOA (0.39) MAOAMAOBMCHR1
SCHEMBL7463814 0.88 PPARG (0.35) MAOAMAOBMCHR1HTR2C
SCHEMBL7458493 0.86 HTR2C (0.39) MAOAMAOBMCHR1HTR2C
SCHEMBL7457048 0.86 MAOB (0.42) MAOAMAOB
SCHEMBL7466444 0.83 HTR2C (0.40) MCHR1HTR2C
SCHEMBL7457982 0.82 MCHR1 (0.30) MCHR1
SCHEMBL7454776 0.80 MCHR1 (0.31) MCHR1
SCHEMBL7465593 0.80
SCHEMBL7465859 0.80 MEN1 (0.30) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed