SCHEMBL7466444

SCHEMBL7466444

Cn1c(C(F)(F)F)cc(=O)n(-c2ccc3snc(COc4ccccc4C(F)(F)F)c3c2)c1=O

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.40
MRGPRX4 Q96LA9 1/20 0.33
RXRA P19793 1/20 0.32
RXRB P28702 1/20 0.32
RXRG P48443 1/20 0.32
HTR2A P28223 2/20 0.32
MCHR1 Q99705 1/20 0.31
SSTR1 P30872 2/20 0.31
SSTR4 P31391 2/20 0.31
KCNH2 Q12809 1/20 0.31
PLK1 P53350 1/20 0.30
GRM4 Q14833 1/20 0.30
MTOR P42345 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455042 0.88 BCAT2 (0.38)
SCHEMBL7457245 0.87 ALDH1A1 (0.37)
SCHEMBL7457982 0.85 MCHR1 (0.30) MCHR1
SCHEMBL7461286 0.84 TACR1 (0.34)
SCHEMBL7454228 0.83 MAOB (0.43) HTR2CMRGPRX4MCHR1
SCHEMBL7459577 0.83 MAOA (0.39) MCHR1KCNH2
SCHEMBL7454776 0.83 MCHR1 (0.31) MCHR1
SCHEMBL7465593 0.83
SCHEMBL7465742 0.83 APP (0.33) HTR2CMCHR1
SCHEMBL7464526 0.83

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed