SCHEMBL7465976

SCHEMBL7465976

CC(C)(C)Cc1cc([N+](=O)[O-])ccc1OC(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
CYP1A2 P05177 2/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
MAPT P10636 2/20 0.41
HPGD P15428 2/20 0.41
ITGA4 P13612 2/20 0.41
ITGB7 P26010 2/20 0.41
MEN1 O00255 4/20 0.40
KMT2A Q03164 4/20 0.40
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
CRHBP P24387 1/20 0.40
HTT P42858 1/20 0.40
CRHR2 Q13324 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7465984 1.00 ALDH1A1 (0.43) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL7465971 0.90 RAB9A (0.41) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL28102381 0.85 ALDH1A1 (0.46) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL32662599 0.84 CYP1A2 (0.46) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL16425424 0.82 TDP1 (0.55) ALDH1A1CYP1A2MAPTHPGDMEN1
SCHEMBL20299855 0.82 BCL9 (0.44) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL8135055 0.82 ALDH1A1 (0.41) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL8135051 0.82 ALDH1A1 (0.41) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL2995979 0.81 CYP1A2 (0.44) ALDH1A1CYP1A2PTGDR2MAPTHPGD
SCHEMBL2993625 0.81 CYP1A2 (0.44) ALDH1A1CYP1A2PTGDR2MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1022277-B1 NEW TAXANE DERIVATIVES YAKULT HONSHA KK (JP) 2002-12-04 EP disclosed
CN-1062561-C 7-halo-and 7 beta, 8 beta-methylene-paclitaxel, antitumor use and pharmaceutical composition containing the same PHARMAIN & UPJOHN CO (US) 2001-02-28 CN disclosed
US-6136808-A ANTITUMOR AGENTS FROM PLANTS KABUSHIKI KAISHA YAKULT HONSHA (JP) 2000-10-24 US disclosed
EP-1022277-A1 NEW TAXANE DERIVATIVES Kabushiki Kaisha Yakult Honsha (JP) 2000-07-26 EP disclosed
CN-1261072-A 7-halogenated and 7 beta, 8 beta-methylene-taxinol, its usage against cancers and medicinal compositions containing it UPJOHN CO (US) 2000-07-26 CN disclosed
CN-1095377-A 7-halo-and 7 beta, 8 beta-methylene-paclitaxel, antitumor use and pharmaceutical composition containing the same UPJOHN CO (US) 1994-11-23 CN disclosed