SCHEMBL7466368

SCHEMBL7466368

Nc1[nH]nc(-c2ccc(F)cc2)c1C(=O)c1cccc(C#CCN2CCOCC2)c1

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 7/20 0.61
GRM5 P41594 1/20 0.40
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
LMNA P02545 1/20 0.37
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
CD274 Q9NZQ7 1/20 0.37
SCN9A Q15858 1/20 0.36
WNT1 P04628 1/20 0.36
DYRK1A Q13627 1/20 0.36
MMP13 P45452 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474820 0.83 ALDH1A1 (0.41) MAPK14ADORA2AADORA1CD274SCN9A
SCHEMBL5322574 0.82 MAPK14 (0.61) MAPK14LMNACD274WNT1DYRK1A
Hydrochloric Acid SCHEMBL7468024 0.81 MAPK14 (0.60) MAPK14MAPK1CD274WNT1DYRK1A
SCHEMBL5321309 0.81 MAPK14 (0.61) MAPK14ADORA2AADORA1
Hydrochloric Acid SCHEMBL7466695 0.80 MAPK14 (0.60) MAPK14ADORA2AADORA1
SCHEMBL7474200 0.80 MAPK14 (0.58) MAPK14GRM5MAPK1
SCHEMBL5321287 0.79 HTR7 (0.47) MAPK14CD274SCN9AWNT1DYRK1A
SCHEMBL7475939 0.77 FKBP1A (0.53) MAPK14LMNARAB9A
SCHEMBL7475479 0.76 MAP3K14 (0.39) MAPK14
SCHEMBL6157440 0.76 MAPK14 (1.00) MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218346-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-07-03 EP disclosed
WO-2001021591-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-29 WO disclosed