SCHEMBL745501

SCHEMBL745501

CC(C)(C)c1ccc(CN(CCc2ccc(Cl)c(Cl)c2)C(=O)c2cccc3c2NCCC3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.39
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
SSTR4 P31391 1/20 0.35
ALDH1A1 P00352 1/20 0.35
SLC13A5 Q86YT5 1/20 0.34
KMT2A Q03164 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
SIGMAR1 Q99720 6/20 0.33
TP53 P04637 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2D6 P10635 2/20 0.33
TSHR P16473 2/20 0.33
ESRRG P62508 2/20 0.33
NR1H4 Q96RI1 1/20 0.33
C5AR1 P21730 1/20 0.33
ESRRB O95718 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL752637 0.99 TMEM97 (0.38) TMEM97OPRM1OPRD1SSTR4ALDH1A1
SCHEMBL749603 0.98 TMEM97 (0.39) TMEM97OPRM1OPRD1SSTR4ALDH1A1
SCHEMBL748523 0.91 LPAR1 (0.38) OPRM1OPRD1SLC13A5KMT2ACRHBP
SCHEMBL748611 0.90 TP53 (0.38) TMEM97OPRM1OPRD1ALDH1A1SLC13A5
SCHEMBL747114 0.90 C5AR1 (0.41) TMEM97OPRM1OPRD1SSTR4SLC13A5
SCHEMBL745512 0.90 OPRM1 (0.34) TMEM97OPRM1OPRD1ALDH1A1KMT2A
SCHEMBL748563 0.90 MBTPS1 (0.39) OPRM1OPRD1SLC13A5KMT2ACRHBP
Hydrochloric Acid SCHEMBL747110 0.89 OPRM1 (0.34) TMEM97OPRM1OPRD1ALDH1A1KMT2A
SCHEMBL746654 0.89 OPRM1 (0.34) TMEM97OPRM1OPRD1ALDH1A1KMT2A
SCHEMBL745473 0.88 KMT2A (0.44) TMEM97OPRM1OPRD1SLC13A5KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US claimed
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed