SCHEMBL7467894

SCHEMBL7467894

Nc1cccc(N)c1-c1nccc(-c2ccncc2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.48
BCR P11274 2/20 0.48
SRC P12931 1/20 0.48
NPC1 O15118 4/20 0.47
GABRA1 P14867 1/20 0.46
GABRG2 P18507 1/20 0.46
GABRB3 P28472 1/20 0.46
GABRA5 P31644 1/20 0.46
GABRA3 P34903 1/20 0.46
HSP90AA1 P07900 2/20 0.44
AURKA O14965 1/20 0.44
PRKACA P17612 1/20 0.44
ADORA2A P29274 1/20 0.44
CYP19A1 P11511 1/20 0.44
KMT2A Q03164 5/20 0.42
CYP1A2 P05177 3/20 0.42
CYP3A4 P08684 3/20 0.42
CYP2D6 P10635 3/20 0.42
CYP2C9 P11712 3/20 0.42
CYP2C19 P33261 3/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467793 0.82 ABL1 (0.45) ABL1BCRSRCNPC1GABRA1
SCHEMBL1231783 0.82 HSP90AA1 (0.64) ABL1BCRSRCHSP90AA1PRKACA
SCHEMBL8501004 0.77 NPC1 (0.70) NPC1GABRA1GABRG2GABRB3GABRA5
SCHEMBL7462995 0.76 KDM4E (0.57) NPC1HSP90AA1CYP19A1KMT2ACYP1A2
SCHEMBL7476570 0.76 KDM4E (0.64) NPC1CYP19A1KMT2ACYP1A2CYP3A4
Ammonia Solution, Strong SCHEMBL27968646 0.75 NPC1 (0.68) NPC1GABRA1GABRG2GABRB3GABRA5
SCHEMBL1891143 0.75 MAPT (0.48) AURKAADORA2AKMT2ACYP1A2CYP3A4
SCHEMBL18905473 0.74 GABRA1 (0.71) NPC1GABRA1GABRG2GABRB3GABRA5
SCHEMBL2684649 0.74 HSP90AA1 (0.70) ABL1BCRSRCNPC1HSP90AA1
SCHEMBL17694969 0.74 NPC1 (0.71) NPC1GABRA1GABRG2GABRB3GABRA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed
EP-0233461-B1 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 1996-03-20 EP disclosed