SCHEMBL7468432

SCHEMBL7468432

Cc1nc(-c2cccc(N)c2)[nH]c1C

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.57
HPGD P15428 4/20 0.57
RAB9A P51151 4/20 0.57
TP53 P04637 3/20 0.57
KDM4E B2RXH2 3/20 0.57
ALDH1A1 P00352 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
PKM P14618 2/20 0.57
MAPT P10636 2/20 0.57
GFER P55789 2/20 0.57
HSD17B10 Q99714 2/20 0.55
PRMT1 Q99873 1/20 0.54
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
POLB P06746 2/20 0.50
HTT P42858 1/20 0.50
USP2 O75604 1/20 0.49
GAA P10253 1/20 0.49
BLM P54132 1/20 0.49
ENPP2 Q13822 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27461517 0.86 NPC1 (0.57) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL28460536 0.82 PIN1 (0.62) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL27461488 0.81 NPC1 (0.52) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL4113640 0.79 PIN1 (0.64) KDM4EALDH1A1GFERGAAPARP1
SCHEMBL7376460 0.79 NPY5R (0.45) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL647088 0.77 PIN1 (0.59) NPC1RAB9AKDM4EMAPTHSD17B10
SCHEMBL23995915 0.77 L3MBTL1 (0.43) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL20425475 0.77 PIN1 (0.66) PARP1PIN1SMPD3
SCHEMBL31398190 0.74 HPGD (0.57) NPC1HPGDRAB9ATP53KDM4E
SCHEMBL1077128 0.74 NPC1 (0.51) NPC1HPGDRAB9ATP53KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216240-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2002-06-26 EP disclosed
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed
WO-2001025229-A1 AMIDE COMPOUNDS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-04-12 WO disclosed