SCHEMBL7468639

SCHEMBL7468639

COc1ccc(Cn2ncnc2CN2CCc3cc(N)ccc3C2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.52
POLB P06746 1/20 0.52
ABCB1 P08183 7/20 0.49
ABCC1 P33527 2/20 0.49
ABCG2 Q9UNQ0 2/20 0.49
DHFR P00374 1/20 0.45
DRD2 P14416 1/20 0.45
KCNH2 Q12809 1/20 0.45
CHRM2 P08172 1/20 0.44
HTR1A P08908 1/20 0.44
CHRM3 P20309 1/20 0.44
DRD4 P21917 1/20 0.44
ADRA1D P25100 1/20 0.44
HTR2C P28335 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
DRD3 P35462 1/20 0.44
HTR2B P41595 1/20 0.44
SLC6A3 Q01959 1/20 0.44
TMEM97 Q5BJF2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6969210 0.85 ABCB1 (0.65) ALDH1A1POLBABCB1ABCC1ABCG2
SCHEMBL7485177 0.84 ALDH1A1 (0.48) ALDH1A1POLBABCB1ABCC1ABCG2
SCHEMBL3156807 0.78 ABCB1 (0.62) ALDH1A1ABCB1ABCC1ABCG2DHFR
SCHEMBL18797822 0.75 SIGMAR1 (0.53) ABCB1ABCC1ABCG2DHFRDRD2
SCHEMBL3157251 0.73 ABCB1 (0.62) ALDH1A1ABCB1ABCC1ABCG2DHFR
SCHEMBL6971135 0.73 SIGMAR1 (0.66) ALDH1A1ABCB1ABCC1ABCG2DRD2
SCHEMBL3296219 0.72 TAAR1 (0.51) ALDH1A1KDM4E
SCHEMBL6962333 0.72 TMEM97 (0.55) ALDH1A1ABCB1ABCC1ABCG2CHRM2
SCHEMBL7480360 0.71 NPBWR1 (0.45) ALDH1A1SIGMAR1KDM4E
SCHEMBL3061384 0.71 CA9 (0.70) ALDH1A1ABCB1ABCC1ABCG2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0902785-B1 PROCESSES AND INTERMEDIATES FOR PREPARING 4'-TRIFLUOROMETHYLBIPHENYL-2-CARBOXYLIC ACID 2-(2H- 1,2,4]TRIAZOL-3-YLMETHYL)-1,2,3,4-TETRAHYDRO-ISOQUINOLIN-6-YL]-AMIDE PFIZER (US) 2002-09-04 EP disclosed
US-5998623-A Process and intermediates for preparing 4'-trifluoromethylbiphenyl-2-carboxylic acid [2-(2H-[1,2,4]triazol-3-ylmethyl)-1,2,3,4-tetrahydro-isoquinolin-6-yl]-a mide PFIZER INC. (US) 1999-12-07 US disclosed