SCHEMBL7469151

SCHEMBL7469151

COc1ccc(-c2nsc3ccc(-n4c(=O)cc(C(F)(F)F)n(C)c4=O)cc23)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPL P05186 1/20 0.37
ALPI P09923 1/20 0.37
CYP1A2 P05177 4/20 0.36
PTGER1 P34995 1/20 0.36
TP53 P04637 2/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CA P42336 1/20 0.35
PIK3CB P42338 1/20 0.35
MTOR P42345 1/20 0.35
PIK3CG P48736 1/20 0.35
PTGS2 P35354 3/20 0.35
PTGS1 P23219 2/20 0.35
FFAR4 Q5NUL3 1/20 0.35
NPC1 O15118 1/20 0.34
PMM2 O15305 1/20 0.34
MIF P14174 1/20 0.34
MPI P34949 1/20 0.34
RAB9A P51151 1/20 0.34
PHOSPHO1 Q8TCT1 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7462871 0.89
SCHEMBL7462316 0.88 ALDH1A1 (0.33) ALPLALPIPTGER1TP53NPC1
SCHEMBL7463075 0.88 TP53 (0.32) TP53PIK3CAMTORNPC1PMM2
SCHEMBL7458904 0.87 PTGS2 (0.36) CYP1A2TP53PTGS2PTGS1MAPT
SCHEMBL7453460 0.87 TP53 (0.35) CYP1A2TP53PTGS2PTGS1MAPT
SCHEMBL7466715 0.83 BRD9 (0.33) TP53
SCHEMBL6770418 0.83 PTGS2 (0.33) MTORPTGS2
SCHEMBL7462604 0.83 ESR1 (0.30)
SCHEMBL7460983 0.82
SCHEMBL6772514 0.82 TGFBR1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0908457-B1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents BASF AG (DE) 2002-11-13 EP disclosed
EP-0908457-A1 3-(1,2-benzisothiazol- and isoxazol-5-Y1)-2,4(1H,3H)-pyrimidinedione or thione and 3-(1,2-benzisothiazol- and isoxazol-5-y1)-4(3H)-pyrimidinone or thione herbicidal agents American Cyanamid Company (US) 1999-04-14 EP disclosed