SCHEMBL7469231

SCHEMBL7469231

CCCCCNc1nc(CC)c(-c2ccc(F)cc2C)nc1CC

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 1/20 0.41
KCNH3 Q9ULD8 1/20 0.39
ACHE P22303 1/20 0.39
CRHR1 P34998 14/20 0.38
HSP90AB1 P08238 2/20 0.38
F2RL1 P55085 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474934 0.86 CRHR1 (0.50) CRHR1
SCHEMBL7477860 0.85 CRHR1 (0.53) KCNH3CRHR1
SCHEMBL6075389 0.78 CRHR1 (0.61) CRHR1
SCHEMBL7481401 0.77 CRHR1 (0.65) CRHR1
SCHEMBL7474850 0.77 CRHR1 (0.46) TLR8ACHECRHR1
SCHEMBL7483586 0.76 TLR8 (0.41) TLR8CRHR1HSP90AB1
SCHEMBL7482439 0.75 CRHR1 (0.53) CRHR1
SCHEMBL7478694 0.74 CRHR1 (0.69) CRHR1
SCHEMBL7481208 0.74 CRHR1 (0.48) KCNH3CRHR1
SCHEMBL7480941 0.73 CRHR1 (0.68) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed