SCHEMBL7474850

SCHEMBL7474850

CCCCCNc1nc(CC)c(-c2ccc(C)cc2C)nc1OC

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 15/20 0.46
TLR8 Q9NR97 2/20 0.39
TLR7 Q9NYK1 1/20 0.39
ACHE P22303 2/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482439 0.89 CRHR1 (0.53) CRHR1
SCHEMBL5533539 0.86 CRHR1 (0.57) CRHR1TLR8TLR7
SCHEMBL7470222 0.83 CRHR1 (0.43) CRHR1TLR8TLR7ACHEPOLB
SCHEMBL7606978 0.82 CRHR1 (0.59) CRHR1
SCHEMBL7481401 0.82 CRHR1 (0.65) CRHR1TLR7POLB
SCHEMBL6204988 0.81 CRHR1 (0.60) CRHR1TLR8TLR7
SCHEMBL7479379 0.81 CRHR1 (0.57) CRHR1
SCHEMBL6202560 0.81 CRHR1 (0.42) CRHR1TLR8TLR7
SCHEMBL7477527 0.80 CRHR1 (0.48) CRHR1TLR8TLR7
SCHEMBL5420383 0.79 CRHR1 (0.68) CRHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1255740-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2002-11-13 EP claimed
WO-2001060806-A2 SUBSTITUTED ARYLPYRAZINES NEUROGEN CORPORATION (US) 2001-08-23 WO claimed