SCHEMBL7469256

SCHEMBL7469256

c1ccc(Nc2nccc(-c3ccnc4ccccc34)n2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 4/20 0.61
CCNB2 O95067 3/20 0.61
CCNB1 P14635 3/20 0.61
CCNB3 Q8WWL7 3/20 0.61
PRKCD Q05655 2/20 0.54
ABL1 P00519 1/20 0.54
EGFR P00533 1/20 0.54
PRKCA P17252 1/20 0.54
KDR P35968 2/20 0.53
PTK2 Q05397 2/20 0.53
PLK1 P53350 1/20 0.53
CDK2 P24941 4/20 0.52
GSK3B P49841 3/20 0.52
CDK4 P11802 3/20 0.52
DYRK1A Q13627 1/20 0.52
CHEK1 O14757 1/20 0.51
IKBKB O14920 1/20 0.51
AURKA O14965 1/20 0.51
NPC1 O15118 1/20 0.51
PDPK1 O15530 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31060885 0.89 CCNB2 (0.62) CDK1CCNB2CCNB1CCNB3KDR
SCHEMBL3605758 0.87 FADS1 (0.62) PRKCDABL1EGFRPRKCAPLK1
SCHEMBL7474541 0.86 RET (0.50) CDK1CCNB2CCNB1CCNB3KDR
SCHEMBL7462357 0.86 CDK1 (0.65) CDK1CCNB2CCNB1CCNB3ABL1
SCHEMBL12783520 0.82 DYRK1A (0.48) CDK1CCNB2CCNB1CCNB3KDR
SCHEMBL31588329 0.76 CCNB2 (0.76) CDK1CCNB2CCNB1CCNB3PRKCD
SCHEMBL144954 0.76 CCNB2 (0.76) CDK1CCNB2CCNB1CCNB3PRKCD
SCHEMBL2544992 0.76 CCNB2 (1.00) CDK1CCNB2CCNB1CCNB3CDK2
SCHEMBL1593016 0.76 PRKCD (0.79) CDK1CCNB2CCNB1CCNB3PRKCD
SCHEMBL27444164 0.76 CDK2 (0.58) CDK1CCNB2CCNB1CCNB3PRKCD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP claimed
EP-0233461-B1 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 1996-03-20 EP claimed
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed