SCHEMBL7474541

SCHEMBL7474541

CCc1ccc(Nc2nccc(-c3ccnc4ccccc34)n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RET P07949 7/20 0.50
BRD4 O60885 2/20 0.50
CDK9 P50750 2/20 0.50
CCNB2 O95067 3/20 0.47
CDK1 P06493 3/20 0.47
CCNB1 P14635 3/20 0.47
CCNB3 Q8WWL7 3/20 0.47
MAPKAPK2 P49137 1/20 0.47
KDR P35968 5/20 0.45
PTK2 Q05397 4/20 0.45
GSK3B P49841 1/20 0.44
PLK1 P53350 2/20 0.44
AURKB Q96GD4 1/20 0.43
AKT1 P31749 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31060885 0.86 CCNB2 (0.62) RETBRD4CDK9CCNB2CDK1
SCHEMBL7469256 0.86 CDK1 (0.61) RETBRD4CDK9CCNB2CDK1
SCHEMBL7467183 0.80 FLT3 (0.60) RETBRD4CDK9CCNB2CDK1
SCHEMBL13185630 0.79 IKBKB (0.60) MAPKAPK2GSK3BPLK1
SCHEMBL7460307 0.78 SYK (0.55)
SCHEMBL7462357 0.78 CDK1 (0.65) RETBRD4CDK9CCNB2CDK1
SCHEMBL12783520 0.77 DYRK1A (0.48) BRD4CDK9CCNB2CDK1CCNB1
SCHEMBL3605758 0.77 FADS1 (0.62) BRD4CDK9PLK1
SCHEMBL7465536 0.74 ABL1 (0.54)
SCHEMBL7475710 0.73 ABL1 (0.71)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed