SCHEMBL7469397

SCHEMBL7469397

CCOC(=O)c1ccc(N2CCC[C@H](Nc3ccccn3)C2)cc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 1/20 0.56
NPC1 O15118 3/20 0.51
RAB9A P51151 2/20 0.51
OPRK1 P41145 1/20 0.50
METAP1 P53582 1/20 0.49
KDM4E B2RXH2 3/20 0.49
MAPT P10636 3/20 0.49
HTT P42858 2/20 0.49
HSD17B10 Q99714 2/20 0.49
ALDH1A1 P00352 2/20 0.49
MAPK1 P28482 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.46
LMNA P02545 1/20 0.45
CHRNA7 P36544 1/20 0.44
CHRNA10 Q9GZZ6 1/20 0.44
CHRNA9 Q9UGM1 1/20 0.44
CASR P41180 1/20 0.43
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7468246 0.90 OPRK1 (0.49) NOS2NPC1RAB9AOPRK1METAP1
SCHEMBL7054705 0.90 OPRK1 (0.49) NOS2NPC1RAB9AOPRK1METAP1
SCHEMBL7461745 0.84 CASR (0.55) NOS2METAP1CASR
SCHEMBL382149 0.83 OPRK1 (0.51) NOS2NPC1RAB9AOPRK1METAP1
SCHEMBL383015 0.83 OPRK1 (0.51) NOS2NPC1RAB9AOPRK1METAP1
SCHEMBL12193435 0.80 NOS2 (0.47) NOS2CHRNA7CHRNA10CHRNA9CASR
SCHEMBL7474418 0.79 NPC1 (0.52) NOS2NPC1RAB9AMETAP1KDM4E
SCHEMBL7466048 0.78 OPRK1 (0.51) NOS2NPC1RAB9AOPRK1KDM4E
SCHEMBL2408945 0.77 CASR (0.54) NOS2METAP1CHRNA7CHRNA10CHRNA9
SCHEMBL382510 0.77 NOS2 (0.51) NOS2OPRK1METAP1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1242409-A2 SUBSTITUTED BISINDOLYLMALEIMIDES F. HOFFMANN-LA ROCHE AG (CH) 2002-09-25 EP disclosed
WO-2001046178-A2 SUBSTITUIERTE BISINDOLYMALEIMIDE F. HOFFMANN-LA ROCHE AG (CH) 2001-06-28 WO disclosed