SCHEMBL7469979

SCHEMBL7469979

COc1ccc(-c2cc(OC(C)C)ccc2Oc2ccc(OCCN3CCCCC3)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 3/20 0.51
ESR1 P03372 8/20 0.51
HRH3 Q9Y5N1 2/20 0.50
KCNH2 Q12809 1/20 0.50
PSMB1 P20618 1/20 0.49
PSMB5 P28074 1/20 0.49
ESR2 Q92731 6/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
MCHR1 Q99705 1/20 0.46
TLR8 Q9NR97 1/20 0.46
TLR7 Q9NYK1 1/20 0.46
KDM4E B2RXH2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7209701 0.85 ESR1 (0.62) LTA4HESR1ESR2
SCHEMBL7778587 0.85 ESR1 (0.63) ESR1HRH3KCNH2ESR2
SCHEMBL7749392 0.83 LTA4H (0.61) LTA4HESR1HRH3KCNH2MCHR1
SCHEMBL7458270 0.78 ESR1 (0.68) ESR1HRH3ESR2
Hydrochloric Acid SCHEMBL5486653 0.77 ESR1 (0.76) ESR1ESR2
SCHEMBL7930070 0.77 ESR1 (0.51) LTA4HESR1ESR2
SCHEMBL7443460 0.76 LTA4H (0.77) LTA4HESR1HRH3KCNH2PSMB1
SCHEMBL14970684 0.76 LTA4H (0.82) LTA4HHRH3PSMB1PSMB5POLB
SCHEMBL15257179 0.76 LTA4H (0.82) LTA4HHRH3PSMB1PSMB5POLB
Hydrochloric Acid SCHEMBL14966283 0.75 LTA4H (0.79) LTA4HHRH3PSMB1PSMB5POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1204655-A2 A CRYSTALLINE FORM OF 6-HYDROXY-3-(4-[2-(PIPERIDIN-1-YL)ETHOXY] PHENOXY)-2-(4-METHOXYPHENYL)BENZO[B]THIOPHENE HYDROCHLORIDE ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2001009115-A2 A NOVEL CRYSTALLINE FORM OF 6-HYDROXY-3- (4-[2-(PIPERIDIN-1- YL)ETHOXY] PHENOXY)-2- (4-METHOXYPHENYL) BENZO[b]THIOPHENE HYDROCHLORIDE ELI LILLY AND COMPANY (US) 2001-02-08 WO disclosed