SCHEMBL7470119

SCHEMBL7470119

O=C(CNC(=O)c1ccc(-c2ccccc2)cc1)NCC(CCCN1CCC(c2ccccc2)CC1)(c1ccccc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 2/20 0.68
SLC6A2 P23975 2/20 0.48
SLC6A4 P31645 2/20 0.48
CCR2 P41597 2/20 0.45
USP5 P45974 2/20 0.44
DRD2 P14416 2/20 0.44
KCNA3 P22001 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
HPGD P15428 1/20 0.41
CD274 Q9NZQ7 1/20 0.41
HTR7 P34969 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRK1 P41145 1/20 0.41
CCR1 P32246 1/20 0.41
CCR3 P51677 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464781 0.94 MCHR1 (0.73) MCHR1CCR2USP5DRD2KCNA3
SCHEMBL7461314 0.93 MCHR1 (0.61) MCHR1SLC6A2SLC6A4CCR2DRD2
SCHEMBL7459547 0.89 MCHR1 (0.65) MCHR1SLC6A2SLC6A4CCR2DRD2
SCHEMBL7459261 0.86 MCHR1 (0.66) MCHR1DRD2KCNA3SIGMAR1HTR7
SCHEMBL7470937 0.85 MCHR1 (0.58) MCHR1SLC6A2SLC6A4CCR2USP5
SCHEMBL7460992 0.85 MCHR1 (0.60) MCHR1SLC6A2SLC6A4CCR2USP5
SCHEMBL7464749 0.85 MCHR1 (0.61) MCHR1SLC6A2SLC6A4CCR2USP5
SCHEMBL7460592 0.84 MCHR1 (0.62) MCHR1SLC6A2SLC6A4DRD2SIGMAR1
SCHEMBL7463548 0.84 MCHR1 (0.60) MCHR1SLC6A2SLC6A4CCR2USP5
SCHEMBL7460278 0.84 MCHR1 (0.71) MCHR1KCNA3SIGMAR1HTR7CCR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1219294-A1 MELANIN CONCENTRATING HORMONE ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-03 EP disclosed
EP-1157003-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS AstraZeneca AB (SE) 2001-11-28 EP disclosed
WO-2000048992-A1 ACYLATED AMINOACETONITRILES AS CYSTEINE PROTEASE INHIBITORS ASTRAZENECA AB (SE) 2000-08-24 WO disclosed