SCHEMBL7470188

SCHEMBL7470188

COC(=O)c1ccc(Cl)cc1NC(=O)NS(=O)(=O)c1ccc[nH]1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRIK1 P39086 5/20 0.45
ALDH1A1 P00352 3/20 0.43
HPGD P15428 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAPT P10636 2/20 0.43
TP53 P04637 2/20 0.43
ABL1 P00519 1/20 0.43
HTT P42858 1/20 0.43
ACLY P53396 1/20 0.42
NR4A2 P43354 2/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7531464 0.87 GRIK1 (0.56) GRIK1
SCHEMBL5166524 0.80 FBP1 (0.49) GRIK1
SCHEMBL3788016 0.79 FLT1 (0.52) ALDH1A1ABL1
SCHEMBL7461264 0.78 FLT1 (0.59) ALDH1A1HPGDMEN1KMT2A
SCHEMBL3782284 0.78 FLT1 (0.48) GRIK1ALDH1A1HPGDMEN1KMT2A
SCHEMBL7461533 0.78 GRIK1 (0.51) GRIK1ALDH1A1HPGDMEN1KMT2A
SCHEMBL7459211 0.77 FLT1 (0.45) ALDH1A1MAPTTP53
SCHEMBL7469556 0.76 TP53 (0.46) GRIK1ALDH1A1HPGDMAPTTP53
SCHEMBL7459021 0.75 FLT1 (0.50) ALDH1A1HPGDMAPTGAA
SCHEMBL3783035 0.73 FLT1 (0.43) GRIK1ALDH1A1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed