SCHEMBL7459211

SCHEMBL7459211

COC(=O)c1ccc(Cl)cc1NC(=O)NS(=O)(=O)c1ccc(-c2cc[nH]n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
FLT1 P17948 9/20 0.45
FLT4 P35916 9/20 0.45
KDR P35968 9/20 0.45
PYGL P06737 1/20 0.43
TP53 P04637 1/20 0.40
MAPT P10636 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
NFKB1 P19838 1/20 0.40
RAB9A P51151 1/20 0.40
NFKB2 Q00653 1/20 0.40
RELA Q04206 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PLA2G2A P14555 1/20 0.39
HRH3 Q9Y5N1 3/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3802745 0.90 GRIK1 (0.47) FLT1FLT4KDRPYGL
SCHEMBL3788016 0.81 FLT1 (0.52) FLT1FLT4KDRPYGLSMN1; SMN2
SCHEMBL7468666 0.81 PYGL (0.44) FLT1FLT4KDRPYGLTP53
SCHEMBL7461264 0.80 FLT1 (0.59) FLT1FLT4KDRALDH1A1LMNA
SCHEMBL7459021 0.78 FLT1 (0.50) FLT1FLT4KDRMAPTSMN1; SMN2
SCHEMBL7470188 0.77 GRIK1 (0.45) TP53MAPTALDH1A1
SCHEMBL3782284 0.76 FLT1 (0.48) FLT1FLT4KDRTP53HRH3
SCHEMBL7461533 0.76 GRIK1 (0.51) FLT1FLT4KDRTP53MAPT
SCHEMBL5166524 0.75 FBP1 (0.49) FLT1FLT4KDR
SCHEMBL7469556 0.74 TP53 (0.46) FLT1FLT4KDRTP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed