SCHEMBL7470896

SCHEMBL7470896

CC(=O)Nc1ccc(Nc2nccc(-c3cccs3)n2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 8/20 0.65
JAK3 P52333 1/20 0.65
NPC1 O15118 3/20 0.59
RAB9A P51151 2/20 0.59
SMN1; SMN2 Q16637 2/20 0.59
ALDH1A1 P00352 1/20 0.59
GAA P10253 1/20 0.59
CYP1A2 P05177 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2C19 P33261 1/20 0.58
MEN1 O00255 3/20 0.57
KMT2A Q03164 3/20 0.57
KDM4E B2RXH2 2/20 0.57
PLK1 P53350 1/20 0.56
IKBKB O14920 1/20 0.52
MAPK1 P28482 1/20 0.51
HSD17B10 Q99714 1/20 0.51
AURKA O14965 1/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HDAC1 Q13547 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11924746 0.88 CYP1A2 (0.61) JAK2JAK3NPC1RAB9ASMN1; SMN2
SCHEMBL8255815 0.83 MAPK8 (0.66) JAK2NPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL7475925 0.82 IKBKB (0.65) JAK2JAK3GAAMEN1KMT2A
SCHEMBL7471621 0.82 MEN1 (0.59) JAK2JAK3NPC1RAB9ASMN1; SMN2
SCHEMBL7475248 0.81 PLK1 (0.58) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL4378143 0.80 JAK2 (0.90) JAK2JAK3GAAMEN1KMT2A
SCHEMBL7466134 0.80 MEN1 (0.62) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL7469184 0.80 SYK (0.54) NPC1RAB9ASMN1; SMN2ALDH1A1GAA
SCHEMBL7470447 0.80 JAK2 (0.79) JAK2JAK3GAAMEN1KMT2A
SCHEMBL3518694 0.79 CCNT1 (0.54) NPC1RAB9ASMN1; SMN2ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed