SCHEMBL7471001

SCHEMBL7471001

Cc1[c]cc(Cl)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 1/20 0.37
NOTUM Q6P988 9/20 0.35
PYCR1 P32322 1/20 0.34
IDO1 P14902 2/20 0.33
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
KDR P35968 1/20 0.33
NPFFR2 Q9Y5X5 1/20 0.33
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31
COMT P21964 1/20 0.31
AR P10275 1/20 0.30
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11263031 0.81 SMN1; SMN2 (0.35) CYP1A2
SCHEMBL455616 0.78 NOTUM (0.33) NOTUM
SCHEMBL7744861 0.78 IDO1 (0.35) RAPGEF4NOTUMIDO1HTR3EHTR3B
SCHEMBL7470531 0.75 IDO1 (0.37) RAPGEF4NOTUMIDO1HTR3EHTR3B
SCHEMBL20562388 0.75 MAPT (0.36) RAPGEF4NOTUMIDO1HTR3EHTR3B
SCHEMBL459052 0.74 PGK1 (0.32)
SCHEMBL2343838 0.72
SCHEMBL2349734 0.71
SCHEMBL3664944 0.71 RAPGEF4 (0.35) RAPGEF4NOTUMIDO1HSD11B1
SCHEMBL27974318 0.71 IDO1 (0.34) NOTUMIDO1HTR3EHTR3BHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1194417-A1 PHENOXY FLUOROPYRIMIDINES BAYER AG (DE) 2002-04-10 EP claimed
WO-2000078733-A1 PHENOXY FLUOROPYRIMIDINES BAYER AKTIENGESELLSCHAFT (DE) 2000-12-28 WO claimed
CN-105143206-B Pyrimidine -2,4- diamine derivative for treating cancer 托马斯·黑勒戴药物研究基金会 2019-01-15 CN disclosed
CN-105143206-A Pyrimidine-2,4-diamine derivatives for treatment of cancer THOMAS HELLEDAYS STIFTELSE F R MEDICINSK FORSKNING 2015-12-09 CN disclosed
EP-1194417-A1 PHENOXY FLUOROPYRIMIDINES BAYER AG (DE) 2002-04-10 EP disclosed
WO-2000078733-A1 PHENOXY FLUOROPYRIMIDINES BAYER AKTIENGESELLSCHAFT (DE) 2000-12-28 WO disclosed