SCHEMBL747155

SCHEMBL747155

CC(C)(C)c1ccc(CN(CCc2ccc(F)cc2)C(=O)c2cc(Cl)cc3c2NCCC3)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
BCL2 P10415 1/20 0.36
ESRRG P62508 2/20 0.35
C5AR1 P21730 1/20 0.34
MCHR1 Q99705 1/20 0.34
PKM P14618 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
F7 P08709 1/20 0.34
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33
SLC2A1 P11166 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL748268 0.99 TP53 (0.38) TP53MAPTBCL2ESRRGC5AR1
SCHEMBL746591 0.92 PARP1 (0.33) TP53MAPTESRRGC5AR1KDM4E
SCHEMBL747946 0.92 TP53 (0.40) TP53MAPTESRRGMCHR1PKM
SCHEMBL751012 0.92 PARP1 (0.36) TP53MAPTBCL2ESRRGC5AR1
Hydrochloric Acid SCHEMBL747648 0.91 PARP1 (0.36) TP53MAPTBCL2ESRRGC5AR1
SCHEMBL747122 0.91 TP53 (0.33) TP53MAPTBCL2ESRRGC5AR1
SCHEMBL748282 0.90 TP53 (0.39) TP53MAPTESRRGMCHR1PKM
Hydrochloric Acid SCHEMBL748492 0.90 TP53 (0.33) TP53MAPTBCL2ESRRGC5AR1
SCHEMBL745512 0.90 OPRM1 (0.34) TP53MAPTESRRGC5AR1PSEN1
SCHEMBL745478 0.90 TP53 (0.38) TP53MAPTESRRGMCHR1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP claimed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US claimed
EP-2049493-B1 COMPOUNDS SUITABLE AS MODULATORS OF HDL CADILA HEALTHCARE LTD (IN) 2012-03-21 EP disclosed
US-8022217-B2 Compounds suitable as modulators of HDL CADILA HEALTHCARE LIMITED (IN) 2011-09-20 US disclosed